13-Tert-Butylergoline Derivatives (original) (raw)
Serotonergic ergoline derivatives
Maria Gioia Fornaretto
Bioorganic & Medicinal Chemistry Letters, 1998
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Synthesis and in vitro structure-activity relationship of 13-tert-butyl-ergoline derivatives as 5-HT1A receptor ligands
Sergio Mantegani
European journal of …, 1997
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Maria Cervini, Mario Varasi, Emanuele Arlandini
European Journal of Medicinal Chemistry, 1999
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Kjell Svensson
Journal of Medicinal Chemistry, 1989
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European Journal of Medicinal Chemistry, 2014
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Electronic Journal of Biomedicine
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Harald Hübner
Bioorganic & Medicinal Chemistry Letters, 1999
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N(1)-substituted ergolines and tryptamines show species differences for the agonist-labeled 5-HT2 receptor
James Audia
European Journal of Pharmacology, 1993
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A Rationale for the Activity Profile of Arylpiperazinylthioalkyls As 5-HT1A-Serotonin and [Alpha] 1-Adrenergic Receptor Ligands
kirti sarbhai
European journal of medicinal chemistry, 2010
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Dopamine/serotonin receptor ligands. Part 17: A cross-target SAR approach: Affinities of azecine-styled ligands for 5-HT2A versus D1 and D2 receptors
Christoph Enzensperger
Bioorganic & Medicinal Chemistry Letters, 2008
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Yunsheng Huang
Bioorganic & Medicinal Chemistry, 2003
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Ergoline Derivatives as a Probe for Featuring the 5-HT 1A Receptor Pharmacophore
Alessandro Dolmella
Journal of Molecular Modeling, 1995
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A New Class of Arylpiperazine Derivatives: the Library Synthesis on SynPhase Lanterns and Biological Evaluation on Serotonin 5-HT 1A and 5-HT 2A Receptors
Maciej Pawłowski
Journal of Combinatorial Chemistry, 2004
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Structure–Activity Relationships of Receptor Binding of 1,4-Dihydropyridine Derivatives
Rahime Şimşek
Biological & Pharmaceutical Bulletin, 2008
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Novel Potent and Selective Central 5-HT 3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT 3 Receptors
Maurizio Anzini
Journal of Medicinal Chemistry, 1999
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Functionally Selective Dopamine D 2 /D 3 Receptor Agonists Comprising an Enyne Moiety
Peter Gmeiner
Journal of Medicinal Chemistry, 2013
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Synthesis and receptor affinities of some conformationally restricted analogues of the dopamine D1 selective ligand (5R)-8-chloro-2,3,4,5-tetrahydro-3-methyl-5-phenyl- 1H-3-benzazepin-7-ol
R. Chipkin, Donald Hou
Journal of medicinal chemistry, 1989
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Influence of N-1 substituent properties on binding affinities of arylpiperazines to the binding site of 5HT1A receptor
Goran Roglic
Journal of The Serbian Chemical Society, 2006
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Design, synthesis and binding properties of novel and selective 5-HT3 and 5-HT4 receptor ligands
Maria Modica
European Journal of Medicinal Chemistry, 2000
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Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1 H -purine-2,6(3 H ,7 H )-dione
Małgorzata Zygmunt, Paweł Żmudzki
Archiv der Pharmazie, 2015
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Synthesis and structure-affinity relationships of novel N-(1-ethyl-4-methylhexahydro-1,4-diazepin-6-yl)pyridine-3-carboxamides with potent serotonin 5-HT3 and dopamine D2 receptor antagonistic activity
Martha Ramirez
2003
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Structure–Activity Relationship and Evaluation of Phenethylamine and Tryptamine Derivatives for Affinity towards 5-Hydroxytryptamine Type 2A Receptor
SHUJIE WANG
Biomolecules & Therapeutics
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Dopamine receptor agonists: 3-allyl-6-chloro-2,3,4,5-tetrahydro-1-(4-hydroxyphenyl)-1H-3-benzazepine-7,8-diol and a series of related 3-benzazepines
Robert Demarinis
Journal of Medicinal Chemistry, 1986
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Synthesis, Biological Evaluation, and Docking Studies of Tetrahydrofuran- Cyclopentanone- and Cyclopentanol-Based Ligands Acting at Adrenergic α 1 - and Serotonine 5-HT 1A Receptors
Silvia Franchini
Journal of Medicinal Chemistry, 2012
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Introduction of a methyl group in α- or β-position of 1-heteroarylethyl-4-phenyl-piperazines affects their dopaminergic/serotonergic properties
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Archiv der Pharmazie, 2001
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Design and Synthesis of Bitopic 2Phenylcyclopropylmethylamine (PCPMA) Derivatives as Selective Dopamine D3 Receptor Ligands
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Synthesis of novel lactam derivatives and their evaluation as ligands for the dopamine receptors, leading to a D 4-selective ligand
Ashraf Abadi
Bioorganic & Medicinal Chemistry, 2007
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(.+-.)-3-Allyl-6-bromo-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine, a new high affinity D1 dopamine receptor ligand: synthesis and structure-activity relationship
John Neumeyer
Journal of Medicinal Chemistry, 1991
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