Serotonergic ergoline derivatives (original) (raw)
Synthesis and in vitro structure-activity relationship of 13-tert-butyl-ergoline derivatives as 5-HT1A receptor ligands
Sergio Mantegani
European journal of …, 1997
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D1 Agonist and/or D2 antagonist dopamine receptor properties of a series of ergoline derivatives: a structure–activity study
Maria Cervini, Mario Varasi, Emanuele Arlandini
European Journal of Medicinal Chemistry, 1999
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Ergoline Derivatives as a Probe for Featuring the 5-HT 1A Receptor Pharmacophore
Alessandro Dolmella
Journal of Molecular Modeling, 1995
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N(1)-substituted ergolines and tryptamines show species differences for the agonist-labeled 5-HT2 receptor
James Audia
European Journal of Pharmacology, 1993
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13-Tert-Butylergoline Derivatives
Maria Gioia Fornaretto
Annals of the New York Academy of Sciences, 1997
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Behavioral studies on LEK-8804, a new ergoline derivative with potent 5-HT1A receptor agonist and 5-HT2 receptor antagonist activity
Igor Krisch
Pharmacology Biochemistry and Behavior, 1994
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6-Methylergoline-8-carboxylic acid esters as serotonin antagonists: N1-substituent effects on 5HT2 receptor affinity
Giff Marzoni
Journal of Medicinal Chemistry, 1987
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Dopamine/serotonin receptor ligands. Part 17: A cross-target SAR approach: Affinities of azecine-styled ligands for 5-HT2A versus D1 and D2 receptors
Christoph Enzensperger
Bioorganic & Medicinal Chemistry Letters, 2008
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A Rationale for the Activity Profile of Arylpiperazinylthioalkyls As 5-HT1A-Serotonin and [Alpha] 1-Adrenergic Receptor Ligands
kirti sarbhai
European journal of medicinal chemistry, 2010
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Receptor binding profiles and quantitative structure–affinity relationships of some 5-substituted-N,N-diallyltryptamines
Paul Daley
Bioorganic & Medicinal Chemistry Letters, 2015
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Azaindole derivatives with high affinity for the dopamine D4 receptor: Synthesis, ligand binding studies and comparison of molecular electrostatic potential maps
Harald Hübner
Bioorganic & Medicinal Chemistry Letters, 1999
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Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1 H -purine-2,6(3 H ,7 H )-dione
Małgorzata Zygmunt, Paweł Żmudzki
Archiv der Pharmazie, 2015
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Guanine nucleotides reveal differential actions of ergot derivatives at D-2 receptors labelled by [3H] spiperone in striatal homogenates
Andrew Gundlach
Brain research, 1983
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INFLUENCE OF ARYLPIPERAZINES AROMATIC STRUCTURE OVER DIFFERENTIAL AFFINITY FOR 5-HT 1A AND 5-HT 2A RECEPTORS
Irene Rebelo
Electronic Journal of Biomedicine
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Resolved 6,7,8,9-tetrahydro-N,N-dimethyl-3H-benz[e]indol-8-amine: central dopamine and serotonin receptor stimulating properties
Kjell Svensson
Journal of Medicinal Chemistry, 1989
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N-(4-Arylpiperazinoalkyl)acetamide derivatives of 1,3- and 3,7-dimethyl-1H-purine-2,6(3H,7H)-diones and their 5-HT6, 5-HT7, and D2 receptors affinity
Paweł Żmudzki
Heterocyclic Communications, 2015
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The synthesis of cyclic and acyclic long-chain arylpiperazine derivatives of salicylamide as serotonin receptor ligands
Piotr kowalski
Journal of Heterocyclic Chemistry, 2008
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A New Class of Arylpiperazine Derivatives: the Library Synthesis on SynPhase Lanterns and Biological Evaluation on Serotonin 5-HT 1A and 5-HT 2A Receptors
Maciej Pawłowski
Journal of Combinatorial Chemistry, 2004
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Receptor binding profiles and QSAR of some 5-substituted-N,N-diallyltryptamines.
Nicholas V Cozzi, Ph.D., Paul Daley
Bioorganic and Medicinal Chemistry Letters, 2016
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Influence of N-1 substituent properties on binding affinities of arylpiperazines to the binding site of 5HT1A receptor
Goran Roglic
Journal of The Serbian Chemical Society, 2006
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Synthesis and structure-affinity relationships of novel N-(1-ethyl-4-methylhexahydro-1,4-diazepin-6-yl)pyridine-3-carboxamides with potent serotonin 5-HT3 and dopamine D2 receptor antagonistic activity
Martha Ramirez
2003
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Ergoline derivatives as highly potent and selective antagonists at the somatostatin sst1 receptor
Thomas Troxler
Bioorganic & Medicinal Chemistry Letters, 2008
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Conformational analysis and theoretical quantitative size and shape-affinity relationships of N< sub> 4-protonated N< sub> 1-arylpiperazine 5-HT< sub> 1A serotoninergic ligands
Marina Cocchi, Maria Cristina Menziani
1997
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Structure–Activity Relationship and Evaluation of Phenethylamine and Tryptamine Derivatives for Affinity towards 5-Hydroxytryptamine Type 2A Receptor
SHUJIE WANG
Biomolecules & Therapeutics
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[14C] - radiolabeling of {[trans-(8β)]-6-methyl-1-(1-methylethyl) ergoline-8-carboxylic acid, 4-methoxycyclohexyl ester (Z)-2-butenedioate [(1:1)]. A potent and selective 5ht2-receptor antagonist
Giff Marzoni
Journal of Labelled Compounds and Radiopharmaceuticals, 1988
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The impact of spacer structure on 5-HT7 and 5-HT1A receptor affinity in the group of long-chain arylpiperazine ligands
Piotr kowalski
Bioorganic & Medicinal Chemistry Letters, 2004
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Bivalent Ligands for the Serotonin 5-HT 3 Receptor
MAURIZIO ANZINI
ACS Medicinal Chemistry Letters, 2011
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