Securinine alkaloids: A new class of GABA receptor antagonist (original) (raw)
Inhibition of [3H]GABA binding to rat brain synaptic membranes by bicuculline related alkaloids
Julianna Kardos
Biochemical Pharmacology, 1984
View PDFchevron_right
(+)-Hydrastine, a potent competitive antagonist at mammalian GABAA receptors
Graham Johnston
British Journal of Pharmacology, 1990
View PDFchevron_right
Bicuculline, an antagonist of GABA and synaptic inhibition in the spinal cord of the cat
Graham Johnston
Brain Research, 1971
View PDFchevron_right
Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor
Joe Steinbach
The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997
View PDFchevron_right
Gaba agonists and antagonists
Graham Johnston
Biochemical Pharmacology, 1979
View PDFchevron_right
Role of cholinergic mechanisms in the mechanism of action of bicuculline
Rita Ostrovskaya
Bulletin of Experimental Biology and Medicine, 1978
View PDFchevron_right
Excitatory amino acid antagonists protect mice against seizures induced by bicuculline
W. Turski
Brain Research, 1990
View PDFchevron_right
Chemical instability of the GABA antagonist bicuculline under physiological conditions
Graham Johnston
Brain Research, 1975
View PDFchevron_right
GABA and bicuculline actions on mouse spinal cord and cortical neurons in cell culture
Linda Nowak
Brain Research, 1982
View PDFchevron_right
Paradoxical anticonvulsant acitivity of the ?hyphen;Aminobutyrate antagonist bicuculline methiodide in the rat striatum
Esper Cavalheiro
Synapse, 1991
View PDFchevron_right
An arylaminopyridazine derivative of gamma-aminobutyric acid (GABA) is a selective and competitive antagonist at the GABAA receptor site
Remy Schlichter
Proceedings of the National Academy of Sciences of the United States of America, 1985
View PDFchevron_right
Action of N-methyl-bicuculline on the binding of γ-aminobutyric acid to a synaptosomal fraction of rat cerebral cortex
Paul Madtes
Experimental Neurology, 1975
View PDFchevron_right
Antagonism between bicuculline and GABA in the cat brain
Graham Johnston
Brain Research, 1971
View PDFchevron_right
5-[1‘-(2‘-N-Arylsulfonyl-1‘,2‘,3‘,4‘-tetrahydroisoquinolyl)]-4,5-dihydro-2(3H)-furanones: Positive Allosteric Modulators of the GABAA Receptor with a New Mode of Action
Rodolphe Razet
Journal of Medicinal Chemistry, 2000
View PDFchevron_right
Bicuculline-insensitive gaba receptors on peripheral autonomic nerve terminals
N. Bowery
European Journal of Pharmacology, 1981
View PDFchevron_right
Bicuculline actions on isolated rat atria, mouse vas-deferens and guinea-pig ileum are unrelated to GABA A receptor blockade
Riccardo Patacchini
General Pharmacology: The Vascular System, 1990
View PDFchevron_right
Neurochemicals for the Investigation of GABAC Receptors
Graham Johnston
Neurochemical Research, 2010
View PDFchevron_right
The epileptogenic action of the taurine analogue guanidinoethane sulfonate may be caused by a blockade of GABA receptors
JM Solis
Journal of Neuroscience Research, 1990
View PDFchevron_right
Studies on the neuropharmacological activity of bicuculline and related compounds
Thomas Miller
Brain Research, 1976
View PDFchevron_right
Antagonists of Ionotropic Receptors for the Inhibitory Neurotransmitter GABA: Therapeutic Indications
Tina Hinton
InTech eBooks, 2018
View PDFchevron_right
Bicuculline-insensitive GABA receptors: studies on the binding of (-)-baclofen to rat cerebellar membranes
Graham Johnston
Neuroscience letters, 1984
View PDFchevron_right
Quantitative evaluation of the potencies of GABA-receptor agonists and antagonists using the rat hippocampal slice preparation
John Kemp
British Journal of Pharmacology, 1986
View PDFchevron_right
N,N′-Dicyclohexylsulfamide and N,N′-diphenethylsulfamide are anticonvulsant sulfamides with affinity for the benzodiazepine binding site of the GABAA receptor and anxiolytic activity in mice
Cristina Wasowski, Valentina Pastore, Luis Bruno-blanch, Andrea Enrique
Biochemical Pharmacology, 2012
View PDFchevron_right
Direct Activation of GABAA Receptors by Loreclezole, an Anticonvulsant Drug with Selectivity for the β-Subunit
Giovanni Biggio
Neuropharmacology, 1996
View PDFchevron_right
Synthesis, Structure−Activity Relationships at the GABA A Receptor in Rat Brain, and Differential Electrophysiological Profile at the Recombinant Human GABA A Receptor of a Series of Substituted 1,2-Diphenylimidazoles
Giovanni Biggio
Journal of Medicinal Chemistry, 2005
View PDFchevron_right
Displacement of [3H]GABA binding to bovine brain receptors by sulfur-containing analogues
Mario Fontana
Neurochemistry International, 1990
View PDFchevron_right
Kinetic differences in GABA receptor binding following GABA and bicuculline methiodide pretreatment
Gabor Maksay
Neuroscience Letters, 1984
View PDFchevron_right
Inhibition of γ-aminobutyric acid uptake by bicuculline analogues
J. Kardos
European journal of …
View PDFchevron_right
A Behavioural and Neurochemical Study in Rats of the Pharmacology of Loreclezole, a Novel Allosteric Modulator of the GABA A Receptor
Mike Snape
Neuropharmacology, 1996
View PDFchevron_right