Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. Synthesis and structure-relationships of α,α-tetrahydropyranylglycine (original) (raw)

Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists

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Bioorganic & Medicinal Chemistry Letters, 2009

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Novel small molecule bradykinin B1 receptor antagonists. Part 1: Benzamides and semicarbazides

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Bioorganic & Medicinal Chemistry Letters, 2010

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Structure activity relationships of non-peptide bradykinin B2 receptor antagonists

Armin Buschauer

Bioorganic & Medicinal Chemistry Letters, 1995

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Structure-based design of six novel classes of nonpeptide antagonists of the bradykinin B2 receptor

Kurt Jarnagin

Bioorganic & Medicinal Chemistry Letters, 2000

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Synthesis and Characterization of Bradykinin B 2 Receptor Agonists Containing Constrained Dipeptide Mimics

Jean-Michel Luccarini

Journal of Medicinal Chemistry, 1999

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Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides

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Journal of Medicinal Chemistry, 2007

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Novel non-peptide lead structures for bradykinin B2-receptor antagonists

Torsten Steinmetzer

Letters in Peptide Science, 2000

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Novel Small Molecule Bradykinin B 2 Receptor Antagonists

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Journal of Medicinal Chemistry, 2009

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2,3-Diaminopyridine as a platform for designing structurally unique nonpeptide bradykinin B1 receptor antagonists

Cuyue Tang

Bioorganic & Medicinal Chemistry Letters, 2005

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Bradykinin B1 antagonists: Biphenyl SAR studies in the cyclopropanecarboxamide series

Christina Marco

Bioorganic & Medicinal Chemistry Letters, 2007

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Aryl sulfonamides containing tetralin allylic amines as potent and selective bradykinin B1 receptor antagonists

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Bioorganic & Medicinal Chemistry Letters, 2010

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In Vitro Pharmacological Profile of a New Small Molecule Bradykinin B2 Receptor Antagonist

anne lesage

Frontiers in Pharmacology, 2020

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Discovery of dihydroquinoxalinone acetamides containing bicyclic amines as potent Bradykinin B1 receptor antagonists

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Bioorganic & Medicinal Chemistry Letters, 2008

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Rationally designed non-peptides: Variously substituted piperazine libraries for the discovery of bradykinin antagonists and other G-protein-coupled receptor ligands

Michael Burkard

Molecular Diversity, 1996

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A new class of bradykinin B1 receptor antagonists with high oral bioavailability and minimal PXR activity

Christina Marco

Bioorganic & medicinal …, 2008

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α-Hydroxy amides as a novel class of bradykinin B1 selective antagonists

Scott Mosser

Bioorganic & Medicinal Chemistry Letters, 2008

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Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profile

Christina Marco

Bioorganic & Medicinal Chemistry Letters, 2008

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Design and Synthesis of New Linear and Cyclic Bradykinin Antagonists

philippe hennig

Journal of Medicinal Chemistry, 1996

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Alpha-hydroxy amides as a novel class of bradykinin B1 selective antagonists

Scott Mosser

Bioorganic & medicinal chemistry letters, 2008

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Synthesis and biological activity of new bradykinin pseudopeptide B1 receptor agonists containing alkylic spacers

Mariella Tancredi

Bioorganic & Medicinal Chemistry Letters, 1997

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A Proposed Model of Bradykinin Bound to the Rat B2 Receptor and Its Utility for Drug Design

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Journal of Medicinal Chemistry, 1994

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New conformationally homogeneous ?-turn antagonists of the human B2 kinin receptor

Andrea Madami

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Aspartic acid scaffold in bradykinin B1 antagonists

Ferenc Bogár, Botond Penke

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2,3-Diaminopyridine Bradykinin B1 Receptor Antagonists

Cuyue Tang

Journal of Medicinal Chemistry, 2004

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The identification of an orally active, nonpeptide bradykinin B 2 receptor antagonist, FR173657

Yoshito Abe

British Journal of Pharmacology, 1997

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Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists

Alessandro Giolitti, Francesca Bellucci

Biochemical Pharmacology, 2004

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3Oxo2-piperazinyl acetamides as potent bradykinin B1 receptor antagonists for the treatment of pain and inflammation

Kevin Yang

International Journal of Food Microbiology, 2011

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