Functional Modulation of a GPCR Conformational Landscape in a Lipid Bilayer (original) (raw)

Structure of a GPCR Ligand in Its Receptor-Bound State: Leukotriene B4 Adopts a Highly Constrained Conformation When Associated to Human BLT2

Eric Guittet

Journal of the American Chemical Society, 2010

View PDFchevron_right

Drug Design for G-Protein-Coupled Receptors by a Ligand-Based NMR Method

Christian Griesinger

Angewandte Chemie International Edition, 2010

View PDFchevron_right

Engineering a G protein-coupled receptor for structural studies: Stabilization of the BLT1 receptor ground state

Michel Laguerre

Protein Science, 2009

View PDFchevron_right

NMR Investigation of Structures of G-protein Coupled Receptor Folding Intermediates

Ismael Mingarro

The Journal of biological chemistry, 2016

View PDFchevron_right

Comparative NMR analysis of an 80-residue G protein-coupled receptor fragment in two membrane mimetic environments

Oliver Zerbe

Biochimica et Biophysica Acta (BBA) - Biomembranes, 2011

View PDFchevron_right

Structural characterization of triple transmembrane domain containing fragments of a yeast G protein-coupled receptor in an organic : aqueous environment by solution-state NMR spectroscopy

Fred Naider

Journal of Peptide Science, 2015

View PDFchevron_right

NMR Structural Studies of Domain 1 of Receptor-associated Protein

M. Migliorini

Journal of Biomolecular NMR, 2000

View PDFchevron_right

Structural insights into positive and negative allosteric regulation of a G protein-coupled receptor through protein-lipid interactions

Jesús Giraldo

Scientific reports, 2018

View PDFchevron_right

Anionic Phospholipids Control Mechanisms of GPCR-G Protein Recognition

Liam Sharp

View PDFchevron_right

How the dynamic properties and functional mechanisms of GPCRs are modulated by their coupling to the membrane environment

Harel Weinstein

Advances in experimental medicine and biology, 2014

View PDFchevron_right

Conformational changes involved in G-protein-coupled-receptor activation

Kenneth A Jacobson

Trends in Pharmacological Sciences, 2008

View PDFchevron_right

Expression, Functional Characterization, and Solid-State NMR Investigation of the G Protein-Coupled GHS Receptor in Bilayer Membranes

Dirk Basson

Scientific Reports, 2017

View PDFchevron_right

Faculty of 1000 evaluation for Ligands and signaling proteins govern the conformational landscape explored by a G protein-coupled receptor

Sebastian Furness

F1000 - Post-publication peer review of the biomedical literature, 2012

View PDFchevron_right

Ligands and signaling proteins govern the conformational landscape explored by a G protein-coupled receptor

Jean-alain Fehrentz

Proceedings of the National Academy of Sciences, 2012

View PDFchevron_right

Influence of Lipid Composition on the Structural Stability of G-Protein Coupled Receptor

Dr. Iqbal Mahmood

Chemical and Pharmaceutical Bulletin, 2013

View PDFchevron_right

Large multiple transmembrane domain fragments of a G protein-coupled receptor: Biosynthesis, purification, and biophysical studies

Fred Naider

Biopolymers, 2012

View PDFchevron_right

Assessing Interactions Between a Polytopic Membrane Protein and Lipid Bilayers Using Differential Scanning Calorimetry and Solid-State NMR

Maureen Leninger

The Journal of Physical Chemistry B, 2018

View PDFchevron_right

Structural basis of G protein-coupled receptor function

John Lloyd

Molecular and Cellular Endocrinology, 1999

View PDFchevron_right

Ligand orientation in a membrane-embedded receptor site revealed by solid-state NMR with paramagnetic relaxation enhancement

Simon G . Patching

Organic & Biomolecular Chemistry, 2015

View PDFchevron_right

Structure of a Double Transmembrane Fragment of a G-Protein-Coupled Receptor in Micelles

Oliver Zerbe

Biophysical Journal, 2009

View PDFchevron_right

Cholesterol Modulates the Membrane Effects and Spatial Organization of Membrane-Penetrating Ligands for G-Protein Coupled Receptors

Harel Weinstein

Biophysical Journal, 2011

View PDFchevron_right

Novel computational methodologies for structural modeling of spacious ligand binding sites of G-protein-coupled receptors: development and application to human leukotriene B4 receptor

Yoko Ishino

TheScientificWorldJournal, 2012

View PDFchevron_right

Structural basis of G protein–coupled receptor–G protein interactions

Joel Karpiak

Nature Chemical Biology, 2010

View PDFchevron_right

New tools for G-protein coupled receptor (GPCR) drug discovery: combination of baculoviral expression system and solid state NMR

Venkata Ratnala

Biotechnology Letters, 2006

View PDFchevron_right

How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape

Sophie MARY

Biochemical Society Transactions, 2013

View PDFchevron_right

Single-molecule view of basal activity and activation mechanisms of the G protein-coupled receptor β 2 AR

Jeffrey Liu

Proceedings of the National Academy of Sciences, 2015

View PDFchevron_right

Correlated motions of conserved polar motifs lay out a plausible mechanism of G protein-coupled receptor activation

Arijit Sarkar

2020

View PDFchevron_right

NMR and computational methods in the structural and dynamic characterization of ligand-receptor interactions

M. Ghitti

2014

View PDFchevron_right

Solid-state NMR and molecular dynamics characterization of cannabinoid receptor-1 (CB1) helix 7 conformational plasticity in model membranes

David Janero

Biochimica et Biophysica Acta (BBA) - Biomembranes, 2009

View PDFchevron_right

Conserved Mechanism of Conformational Stability and Dynamics in G-Protein-Coupled Receptors

sangbae lee

Journal of Chemical Theory and Computation, 2016

View PDFchevron_right

Structural studies of fragments of G-protein coupled receptors and their ligands by NMR

Alexey Neumoin

2009

View PDFchevron_right

Solution- and solid-state NMR studies of GPCRs and their ligands

Alan Goddard

Biochimica et Biophysica Acta (BBA) - Biomembranes, 2011

View PDFchevron_right