Comparative Inhibition of Voltage-Gated Cation Channels by Local Anesthetics (original) (raw)

Mechanisms of use-dependent block of sodium channels in excitable membranes by local anesthetics

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Molecular and kinetic determinants of local anaesthetic action on sodium channels

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Molecular mechanism of allosteric modification of voltage-dependent sodium channels by local anesthetics

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Selective Interaction of Local Anesthetics with a Peptide Derived from the Voltage-Gated Na+ Channel

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Block of Inactivation-deficient Na+ Channels by Local Anesthetics in Stably Transfected Mammalian Cells

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Bupivacaine Blocks N-Type Inactivating Kv Channels in the Open State: No Allosteric Effect on Inactivation Kinetics

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Binding of General Anesthetics to Ion Channels

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Kinetic analysis of phasic inhibition of neuronal sodium currents by lidocaine and bupivacaine

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Interaction of local anesthetics with the K⁺channel pore domain

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Novel Molecular Determinants in the Pore Region of Sodium Channels Regulate Local Anesthetic Binding

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Membrane-Mediated Activity of Local Anesthetics

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Ketamine blockade of voltage-gated sodium channels: evidence for a shared receptor site with local anesthetics

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Structural and gating changes of the sodium channel induced by mutation of a residue in the upper third of IVS6, creating an external access path for local anesthetics

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Local anesthetic properties of opioids and phencyclidines: Interaction with the voltage-dependent, batrachotoxin binding site in sodium channels

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Local Anesthetic Neurotoxicity Does Not Result from Blockade of Voltage-Gated Sodium Channels

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Sodium channel selectivity filter regulates antiarrhythmic drug binding

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The sensitivity of sodium channels in immature and mature rat CA1 neurones to the local anaesthetics procaine and lidocaine

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Identification of a critical binding site for local anaesthetics in the side pockets of K v 1 channels

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Effects of general anaesthetics on neuronal sodium and potassium channels

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Comparative Inhibition of Voltage-Gated Cation Channels by Local Anesthetics (original) (raw)

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