Synthesis of 4-hydroxy-2-methylproline derivatives via pyrrolidine ring assembly: chromatographic resolution and diastereoselective synthesis approaches (original ) (raw )General strategy for a short and efficient synthesis of 3-hydroxy-4-methylprolines (HMP)
Debendra Mohapatra
Tetrahedron Letters, 2006
View PDFchevron_right
A stereodivergent route to two epimeric 2-pyrrolidinylglycine derivatives
Ayan Bandyopadhyay
Tetrahedron Letters, 2009
View PDFchevron_right
Stereoselective pyrrolidine synthesis and approaches to cyclic tetrapeptides
Nabaz salih
2015
View PDFchevron_right
Stereoselective syntheses of 3-mercaptoproline derivatives protected for solid phase peptide synthesis
Steve Kolodziej
International Journal of Peptide and Protein Research, 1996
View PDFchevron_right
Diastereoselective Synthesis of 5-Heteroaryl-Substituted Prolines Useful for Controlling Peptide-Bond Geometry
Rafat Ali
Organic letters, 2016
View PDFchevron_right
Concise, Stereoselective Route to the Four Diastereoisomers of 4-Methylproline
Murray Munro
Journal of Natural Products, 2008
View PDFchevron_right
Direct access to side chain N,N′-diaminoalkylated derivatives of basic amino acids suitable for solid-phase peptide synthesis
Predrag Cudic
Amino Acids, 2013
View PDFchevron_right
Synthesis of di-and trihydroxy proline derivatives from D-glycals: Application in the synthesis of polysubstituted pyrrolizidines and bioactive 1C-aryl/alkyl pyrrolidines
Sateesh Dubbu
Carbohydrate Research, 2019
View PDFchevron_right
Straightforward synthesis of enantiopure 2-aminomethyl and 2-hydroxymethyl pyrrolidines with complete stereocontrol
Stefano Cicchi
Tetrahedron letters, 2005
View PDFchevron_right
ChemInform Abstract: Aspartimide Formation in Peptide Chemistry: Occurrence, Prevention Strategies and the Role of N‐Hydroxylamines
Ayman El-Faham
ChemInform, 2012
View PDFchevron_right
Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides
Walter Cabri
ACS Sustainable Chemistry & Engineering, 2019
View PDFchevron_right
Synthesis of ω-Oxo Amino Acids and trans-5-Substituted Proline Derivatives Using Cross-Metathesis of Unsaturated Amino Acids
Nabaz salih
The Journal of organic chemistry, 2016
View PDFchevron_right
Three-Component Synthesis of Polysubstituted Homoproline Analogs
Konstantin Kudryavtsev , Константин Кудрявцев
Molecules, 2005
View PDFchevron_right
Peptides derived from α-hydroxymethylserine: Aspects of solid-phase synthesis
Marcin Stasiak
Letters in Peptide Science, 1998
View PDFchevron_right
Aspartimide formation in peptide chemistry: occurrence, prevention strategies and the role of N-hydroxylamines
Ayman El-Faham
Tetrahedron, 2011
View PDFchevron_right
A straightforward route to enantiopure 2-substituted-3,4-dehydro-β-proline via ring closing metathesis
Alessandra Tolomelli , Luca Gentilucci
Amino Acids, 2011
View PDFchevron_right
1,3-Dichloroacetone: A Robust Reagent for Preparing Bicyclic Peptides
Qingqing Lin
ACS Omega, 2020
View PDFchevron_right
The synthesis of ‘difficult’ peptides using 2-hydroxy-4-methoxybenzyl or pseudoproline amino acid building blocks: a comparative study
Nicholas Ede
Journal of Peptide Science, 1999
View PDFchevron_right
S-2,4,6-trimethoxybenzyl (Tmob): a novel cysteine protecting group for the N.alpha.-(9-fluorenylmethoxycarbonyl) (Fmoc) strategy of peptide synthesis
George Barany
The Journal of Organic Chemistry, 1992
View PDFchevron_right
Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis of C-Terminal-Modified and Cyclic Peptides 1 , 2 , 3
Josef Vagner
Journal of the American Chemical Society, 1998
View PDFchevron_right
Enantioselective Solid-Phase Peptide Synthesis Using Traceless Chiral Coupling Reagents and Racemic Amino Acids
Beata Kolesińska
Helvetica Chimica Acta, 2012
View PDFchevron_right
Stereoselective Syntheses of 4-Oxa Diaminopimelic Acid and Its Protected Derivatives via Aziridine Ring Opening
Hongqiang Liu
Organic Letters, 2007
View PDFchevron_right
An Improved Procedure for N- to C-Directed (Inverse) Solid-Phase Peptide Synthesis
Gunnar Lindeberg
Journal of Combinatorial Chemistry, 2000
View PDFchevron_right
3,4-Disubstituted .gamma.-lactam rings as conformationally constrained mimics of peptide derivatives containing aspartic acid or norleucine
David Garvey
The Journal of Organic Chemistry, 1990
View PDFchevron_right
Synthesis of enantiomerically pure delta-benzylproline derivatives
Isabel Rodriguez
New J. Chem., 2015
View PDFchevron_right
Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis of C-Terminal-Modified and Cyclic Peptides1 , 2 , 3
George Barany
Journal of the American Chemical Society, 1998
View PDFchevron_right
Routes to 4-substituted analogues of the glycine/NMDA antagonist HA-996. Enantioselective synthesis of (3R,4R) 3-amino-1-hydroxy-4-methyl-2-pyrrolidinone (L-687, 414)
Paul D Leeson
Tetrahedron, 1992
View PDFchevron_right
2-Amino-4-pyrrolidinothieno[2,3- d ]pyrimidine-6-carboxylic Acid as an N -Terminal Surrogate in Amino Acid and Peptide Analogues
Vassiliki Magafa
Synthesis, 2005
View PDFchevron_right
Methods of the site-selective solid phase synthesis of peptide-derived Amadori products
Katarzyna Kapczyńska
Amino Acids, 2010
View PDFchevron_right
Organocatalytic Activation of Diethyl Glutaconate for the Diastereo- and Enantioselective Assembly of NH-Free 2,3,4-Trisubstituted Pyrrolidines
jean paul rodriguez
Organic letters, 2017
View PDFchevron_right
2-(2,4-DINITROPHENYL)ETHYLOXYCARBONYL-AMINO Acids, New Base Labile Protected Derivatives Suitable for Solid-Phase Peptide Synthesis
Ramon Eritja
Tetrahedron Letters, 1992
View PDFchevron_right
Highly Stereoselective Syntheses of Proline-Derived Vicinal Amino Alcohols through Grignard Addition onto N-Tosylprolinal
Saikat Chaudhuri
Synlett, 2015
View PDFchevron_right
Diastereoselective synthesis of syn,syn- and syn,anti-2,4-diamino-3-hydroxyglutaric acid derivatives from ethyl α-acyl alaninates
AURELIO GARCIA CSAKY
Tetrahedron, 1999
View PDFchevron_right
2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis
Ayman El-Faham
Amino acids, 2015
View PDFchevron_right
Solid-phase synthesis of peptide-4-nitroanilides
Angelika Schierhorn , Mike Schutkowski
International Journal of Peptide and Protein Research, 1996
View PDFchevron_right