Dalargin and [Cys-(O2NH2)]2 analogues of enkephalins and their selectivity for μ opioid receptors (original) (raw)
[D-Ala2,Leu5,Cys6]enkephalin: Short-term agonist effects and long-term antagonism at delta opioid receptors
Daniel Calcagnetti
Peptides, 1989
View PDFchevron_right
Systemic analgesic activity and .delta.-opioid selectivity in [2,6-dimethyl-Tyr1, D-Pen2, D-Pen5]enkephalin
Henry I. Mosberg
Journal of Medicinal Chemistry, 1992
View PDFchevron_right
Pharmacological and functional biochemical properties of d-Ala2-d-Nle5-enkephalin-Arg-Phe
Judit Farkas
Regulatory Peptides, 2004
View PDFchevron_right
Irreversible labelling of rat brain opioid receptors by enkephalin chloromethyl ketones
Mária Wollemann, Mária Szücs
Neuropeptides, 1986
View PDFchevron_right
Studies on spinal opiate receptor pharmacology. III. Analgetic effects of enkephalin dimers as measured by cutaneous-thermal and visceral-chemical evoked responses
David Rodbard
Brain Research, 1985
View PDFchevron_right
Antinociceptive activity of glycosidic enkephalin analogues
Gregorio Valencia
Psychopharmacology, 1990
View PDFchevron_right
Differences in physical dependence induced by selective μ or δ opioid agonists and by endogenous enkephalins protected by peptidase inhibitors
R. Maldonado
Brain Research, 1990
View PDFchevron_right
DOCKING STUDIES OF SELECTIVE ENKEPHALIN ANALOGUES TO DELTA-OPIOID RECEPTOR
Nevena Pencheva, Tatyana Dzimbova
bioinfo.swu.bg
View PDFchevron_right
к-Opioid receptor stimulation abolishes μ- but not δ-mediated inhibitory control of spinal Met-enkephalin release
E. Collin
Neuroscience Letters, 1992
View PDFchevron_right
Different Regulation of Human δ-Opioid Receptors by SNC-80 [(+)-4-[(αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N,N-diethylbenzamide] and Endogenous Enkephalins
stephane allouche
Journal of Pharmacology and Experimental Therapeutics, 2004
View PDFchevron_right
A novel cyclic enkephalin analogue with potent opioid antagonist activity
Peter Schiller
Bioorganic & Medicinal Chemistry Letters, 2004
View PDFchevron_right
Ring substituted and other conformationally constrained tyrosine analogs of [cyclic] [D-Pen2,D-Pen5]enkephalin with .delta.-opioid receptor selectivity
Victor Hruby
Journal of Medicinal Chemistry, 1992
View PDFchevron_right
A cyclic enkephalin analog with high in vitro opiate activity
Peter Schiller
Proceedings of the National Academy of Sciences, 1980
View PDFchevron_right
Novel approaches in the development of new analgesics
Pascale Coric, Serge Turcaud
Neurophysiologie Clinique/Clinical Neurophysiology, 1990
View PDFchevron_right
Facilitation of enkephalins catabolism inhibitor-induced antinociception by drugs classically used in pain management
Bernard Roques, Jesùs Benavides
Neuropharmacology, 2001
View PDFchevron_right
Cyclic Enkephalin Analogues with Exceptional Potency and Selectivity for δ-Opioid Receptors 1
Victor Hruby is to
Journal of Medicinal Chemistry, 1997
View PDFchevron_right
Opioid enhancement of evoked [Met5]enkephalin release requires activation of cholinergic receptors: possible involvement of intracellular calcium
Alan Gintzler
Proceedings of the National Academy of Sciences, 1992
View PDFchevron_right
Effects of Opioids on Noncholinergic Excitatory Responses of the Guinea-Pig Isolated Ileum: Inhibition of Release of Enteric Substance P
Alan Gintzler
British Journal of Pharmacology, 1982
View PDFchevron_right
Naltrindole, an opioid δ antagonist, blocks the enhancement of morphine-antinociception induced by a CCKB antagonist in the rat
Michael Ossipov
Neuroscience Letters, 1994
View PDFchevron_right
Cyclic enkephalin analogs with exceptional potency at peripheral .delta. opioid receptors
Victor Hruby is to
Journal of Medicinal Chemistry, 1994
View PDFchevron_right
Bis-penicillamine enkephalins possess highly improved specificity toward delta opioid receptors
Victor Hruby is to
Proceedings of the National Academy of Sciences, 1983
View PDFchevron_right
Cyclic Enkephalin Analogues with Exceptional Potency and Selectivity for δ-Opioid Receptors
Victor Hruby
Journal of Medicinal Chemistry, 1997
View PDFchevron_right
Pharmacological properties of a proenkephalin A-derived opioid peptide: BAM 18
Diana E Hurlbut
European Journal of Pharmacology, 1987
View PDFchevron_right
Irreversible labelling of the opioid receptors by a melphalan-substituted [Met5]enkephalin-Arg-Phe derivative
Anna Borsodi, Gyorgy Orosz
European Journal of Pharmacology, 1999
View PDFchevron_right
Stimulation of ?Opioid Receptors Reduces the In Vivo Binding of the Cholecystokinin (CCK)-B-Selective Agonist [ 3 H]pBC 264: Evidence for a Physiological Regulation of CCKergic Systems by Endogenous Enkephalins
Christiane Durieux
Journal of Neurochemistry, 1992
View PDFchevron_right
Comparing analgesia and μ-opioid receptor internalization produced by intrathecal enkephalin: requirement for peptidase inhibition
Orlando Perez
View PDFchevron_right
Autoradiographic localization of δ opioid receptors in the rat brain using a highly selective bis-penicillamine cyclic enkephalin analog
Sue Duckles
Eur J Pharmacol, 1985
View PDFchevron_right