Structure–affinity relationships of the affinity of 2-pyrazolyl adenosine analogues for the adenosine A2A receptor (original) (raw)
Synthesis and biological data of 4-amino-1-(2-chloro-2-phenylethyl)-1 H-pyrazolo[3,4- b]pyridine-5-carboxylic acid ethyl esters, a new series of A 1-adenosine receptor (A 1AR) ligands
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Bioorganic & Medicinal Chemistry, 2004
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Comparative molecular field analysis of selective A< sub> 3 adenosine receptor agonists
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1995
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2-Substituted adenosine derivatives: affinity and efficacy at four subtypes of human adenosine receptors
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Biochemical Pharmacology, 2004
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Bioorganic & Medicinal Chemistry Letters, 1997
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Structure−Activity Relationships of 2, N 6 ,5‘-Substituted Adenosine Derivatives with Potent Activity at the A 2B Adenosine Receptor
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Journal of Medicinal Chemistry, 2007
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Pyrazolo [4, 3-e]-1, 2, 4-triazolo [1, 5-c] pyrimidine derivatives as adenosine receptor antagonists. Influence of the N5 substituent on the affinity at the human A3 and …
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Journal of medicinal …, 2003
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Bioorganic & Medicinal Chemistry Letters, 2011
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Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines
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2014
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Water-Soluble Pyrazolo[4,3- e ][1,2,4]triazolo[1,5- c ]pyrimidines as Human A 3 Adenosine Receptor Antagonists
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Journal of Medicinal Chemistry, 2012
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Philip van Galen
European Journal of Pharmacology: Molecular Pharmacology, 1989
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Introduction of alkynyl chains on C-8 of adenosine led to very selective antagonists of the A3 adenosine receptor
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Bioorganic & Medicinal Chemistry Letters, 2001
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N 6-Cycloalkyl-and N 6-Bicycloalkyl-C 5′(C 2′)-modified Adenosine Derivatives as High-Affinity and Selective Agonists at the Human A1 Adenosine Receptor with …
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Journal of medicinal …, 2009
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Bioorganic & Medicinal Chemistry, 2011
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5′-Carbamoyl derivatives of 2′-C-methyl-purine nucleosides as selective A1 adenosine receptor agonists: Affinity, efficacy, and selectivity for A1 receptor from different species
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