Investigation of the effects of drugs effective on PI3K-AKT signaling pathway in colorectal cancer alone and in combination (original) (raw)

The Dual PI3K/mTOR Inhibitor NVP-BEZ235 Induces Tumor Regression in a Genetically Engineered Mouse Model of PIK3CA Wild-Type Colorectal Cancer

Wei Chen

PLoS ONE, 2011

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233 Inhibition of PI3K as a potential treatment for cancer

Ana Carrera

European Journal of Cancer Supplements, 2010

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NVP-BEZ235, a Dual PI3K/mTOR Inhibitor, Prevents PI3K Signaling and Inhibits the Growth of Cancer Cells with Activating PI3K Mutations

Serena Di Cosimo

Cancer Research, 2008

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The efficacy of a novel, dual PI3K/mTOR inhibitor NVP-BEZ235 to enhance chemotherapy and antiangiogenic response in pancreatic cancer

Margaret Schwarz

Journal of Cellular Biochemistry, 2012

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The novel dual PI3K/mTOR inhibitor NVP-BGT226 displays cytotoxic activity in both normoxic and hypoxic hepatocarcinoma cells

Ayman Alameen, Giorgio Zauli, Carolina Simioni

Oncotarget, 2015

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Supplementary Materials, Tables 1-2, Figure Legends 1-8 from Identification and Characterization of NVP-BKM120, an Orally Available Pan-Class I PI3-Kinase Inhibitor

Tobi Nagel

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PI3K/Akt and GSK-3β prevents in a differential fashion the malignant phenotype of colorectal cancer cells

José Morgado-díaz

Journal of Cancer Research and Clinical Oncology, 2010

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Identification of NVP-BKM120 as a Potent, Selective, Orally Bioavailable Class I PI3 Kinase Inhibitor for Treating Cancer

Thomas Hendrickson

ACS Medicinal Chemistry Letters, 2011

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Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor

David Cebrian

Bioorganic & Medicinal Chemistry Letters, 2012

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The dual PI3K/mTOR inhibitor NVP-BEZ235 enhances nab-paclitaxel antitumor response in experimental gastric cancer

Margaret Schwarz

International Journal of Oncology, 2013

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Identification and Characterization of NVP-BKM120, an Orally Available Pan-Class I PI3-Kinase Inhibitor

Tobi Nagel

Molecular Cancer Therapeutics, 2012

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The synergistic anti-proliferative effect of the combination of diosmin and BEZ-235 (dactolisib) on the HCT-116 colorectal cancer cell line occurs through inhibition of the PI3K/Akt/mTOR/NF-κB axis

Rana Elmahdy

Molecular Biology Reports, 2020

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New Potent and Selective Inhibitor of Pim-1/3 Protein Kinases Sensitizes Human Colon Carcinoma Cells to Doxorubicin

Shuguang Liang

Anti-Cancer Agents in Medicinal Chemistry, 2014

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Synergistic antitumor effect of NVP-BEZ235 and CAPE on MDA-MB-231 breast cancer cells

Nafiseh Esmaeil

Biomedicine & Pharmacotherapy, 2017

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IN SILICO STUDIES OF INDAZOLE PYRIDINE ANALOGS AS POTENT INHIBITORS OF AKT PROTEIN IN CANCER

Manoj Kumar

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Carcinogenesis of PIK3CA

Tooba Anum

Hereditary Cancer in Clinical Practice, 2013

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Farelerde AK27 Bitkisel Karışımının Ehrlich Ascites Karsinoma Üzerine Antitümorijenik Etkisi

İbrahim KiliÇ

Kafkas Universitesi Veteriner Fakultesi Dergisi

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Cancer Therapy : Preclinical Dual Targeting of Phosphoinositide 3-Kinase and Mammalian Target of Rapamycin Using NVP-BEZ 235 as a Novel Therapeutic Approach in Human Ovarian Carcinoma

Amer Karam

2011

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Phytochemicals and PI3K Inhibitors in Cancer-An Insight

tabassum khan

Frontiers in pharmacology, 2017

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Activity of any class IA PI3K isoform can sustain cell proliferation and survival

Bart Vanhaesebroeck

Proceedings of the National Academy of Sciences, 2010

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Characterization of the Activity of the PI3K/mTOR Inhibitor XL765 (SAR245409) in Tumor Models with Diverse Genetic Alterations Affecting the PI3K Pathway

Chris Buhr, Artur Plonowski

Molecular Cancer Therapeutics, 2014

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Therapeutic Potency of PI3K Pharmacological Inhibitors of Gastrointestinal Cancer

Maliheh Moradzadeh

Middle East Journal of Digestive Diseases, 2018

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Discovery of novel anticancer therapeutics targeting the PI3K/Akt/mTOR pathway

Pascal Furet

Future Medicinal Chemistry, 2009

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Selective Eradication of Colon Cancer Cells Harboring PI3K and/or MAPK Pathway Mutations in 3D Culture by Combined PI3K/AKT/mTOR Pathway and MEK Inhibition

Helmut Dolznig

International Journal of Molecular Sciences

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Nitrik Oksit Sentaz (NOS) İnhibitörlerinin Sıçanlarda Çok Düşük Frekanslı Manyetik Alanın İndüklediği Analjezi Üzerine Etkileri

Ercan Ozdemir

Genel Tip Dergisi, 2017

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Potent Inhibitors of Phosphatidylinositol 3 (PI3) Kinase that have Antiproliferative Activity Only When Delivered as Prodrug Forms

SYAZWANI ITRI BINTI AMRAN FBME A

ChemMedChem, 2013

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