original ) (raw )Molecular Recognition of Sub-micromolar Inhibitors by the Epinephrine-Synthesizing Enzyme Phenylethanolamine N- Methyltransferase
Fiona McMillan
Journal of Medicinal Chemistry, 2004
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Evaluation of the Abuse Potential of Novel Amphetamine Derivatives with Modifications on the Amine (NBNA) and Phenyl (EDA, PMEA, 2-APN) Sites
Raly James Custodio
Biomolecules & Therapeutics, 2017
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Heterocyclic cycloalkanol ethylamines as norepinephrine reuptake inhibitors
Yingru Zhang
Bioorganic & Medicinal Chemistry Letters, 2010
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Analytical characterization of four new ortho -methoxybenzylated amphetamine-type designer drugs
Folker Westphal
Drug Testing and Analysis, 2015
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Comparative molecular field analysis (CoMFA) models of phenylethanolamine N-methyltransferase (PNMT) and the α2-adrenoceptor: The development of new, highly selective inhibitors of PNMT
Ravi Jalluri
Bioorganic & Medicinal Chemistry Letters, 1999
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Receptor interaction profiles of novel N-2-methoxybenzyl (NBOMe) derivatives of 2,5-dimethoxy-substituted phenethylamines (2C drugs)
Marius C Hoener
Neuropharmacology, 2015
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Noncompetitive inhibition of indolethylamine-N-methyltransferase by N,N-dimethyltryptamine and N,N-dimethylaminopropyltryptamine.
Nicholas V Cozzi, Ph.D.
Biochemistry, 2014
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Chromophoric Derivatives of Amphetamine Analogues: Strucutural Characterization by Electron Impact Mass Spectrometry
F. Castagna
Organic Mass Spectrometry, 1992
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Naphthylisopropylamine and N-benzylamphetamine derivatives as monoamine oxidase inhibitors
Bruce Cassels
Bioorganic & Medicinal Chemistry, 2009
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Synthesis of some novel potent and selective catechol O-methyltransferase inhibitors
Jarmo Pystynen
Journal of Medicinal Chemistry, 1989
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Enzymatic enantiomeric resolution of phenylethylamines structurally related to amphetamine
Pilar Bosch
Organic & biomolecular chemistry, 2011
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Synthesis and pharmacological examination of benzofuran, indan, and tetralin analogues of 3,4-(methylenedioxy)amphetamine.
Nicholas V Cozzi, Ph.D.
Journal of Medicinal Chemistry, 1993
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Effects of Methylphenidate Analogues on Phenethylamine Substrates for the Striatal Dopamine Transporter
Howard Deutsch
Journal of Neurochemistry, 2008
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Noncompetitive Inhibition of Indolethylamine N-Methyltransferase by N,N Dimethyltryptamine (DMT) and N,N-Dimethylaminopropyltryptamine
Timur Mavlyutov
Biochemistry, 2014
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Pharmacological Characterization of 4-Methylthioamphetamine Derivatives
Ramón Sotomayor-zárate
Molecules
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Inhibition of transport function and desipramine binding at the human noradrenaline transporter by N-ethylmaleimide and protection by substrate analogs.
Nicholas V Cozzi, Ph.D.
Naunyn-Schmiedeberg's Archives of Pharmacology, 2002
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Stereospecific inhibition of monoamine uptake transporters by meta-hydroxyephedrine isomers.
Nicholas V Cozzi, Ph.D. , Marcian Van Dort , Arnold Ruoho
Journal of Neural Transmission, 2002
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Quantum mechanical conformational analysis of heterocyclic analogues of norephedrine
J. Kaneti
Chemico-Biological Interactions, 1980
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Structure−Activity Relationship Studies of 4-[2-(Diphenylmethoxy)ethyl]-1-benzylpiperidine Derivatives and Their N-Analogues: Evaluation of Behavioral Activity of O- and N-Analogues and Their Binding to Monoamine Transporters
aloke dutta
Journal of Medicinal Chemistry, 2001
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Monoamine Oxidase Inhibitory Properties of Some Methoxylated and Alkylthio Amphetamine Derivatives
Fabio Sparatore
Biochemical Pharmacology, 1997
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Binding and functional affinity of some newly synthesized phenethylamine and phenoxypropanolamine derivatives for their agonistic activity at recombinant human β 3 -adrenoceptor
maruf ahmed
Journal of Pharmacy and Pharmacology, 2003
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Conformational analysis of amphetamine in solution based on unambiguous assignment of the diastereotopic benzylic protons in the 1H NMR spectra
James Knittel
Tetrahedron Letters, 1981
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Comparative potencies of 3,4-methylenedioxymethamphetamine (MDMA) analogues as inhibitors of [3 H]noradrenaline and [3 H]5-HT transport in mammalian cell lines
therese montgomery
British Journal of Pharmacology, 2009
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The influence of R and S configurations of a series of amphetamine derivatives on quantitative structure–activity relationship models
Márcia Miguel Castro Ferreira
Analytica Chimica Acta, 2013
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Resolved pyrrolidine, piperidine, and perhydroazepine analogs of the muscarinic agent N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide
Patrizia Caldirola
Journal of Medicinal Chemistry, 1990
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Structure–Activity Relationship and Evaluation of Phenethylamine and Tryptamine Derivatives for Affinity towards 5-Hydroxytryptamine Type 2A Receptor
SHUJIE WANG
Biomolecules & Therapeutics
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Adeboye Adejare
Chemical Biology & Drug Design, 2011
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Biochemical and Behavioral Characterization of Novel Methylphenidate Analogs
Heidy Pacheco
Journal of Pharmacology and Experimental Therapeutics, 2002
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Conformationally restrained analogues of sympathomimetic catecholamines
Elisabetta Orlandini
European Journal of Medicinal Chemistry, 2002
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Structure− Activity Relationships for a Series of Bis (phenylalkyl) amines: Potent Subtype-Selective Inhibitors of N-Methyl-d-aspartate Receptors
C. Sansom
J. Med. …, 1998
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Monoamine oxidase inhibitory effects of some 4-aminophenethylamine derivatives
Federico Dajas
Biochemical Pharmacology, 1994
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Microdialysis studies on 3,4-methylenedioxyamphetamine and structurally related analogues
David Nichols
European Journal of Pharmacology, 1991
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Synthesis and structureâaffinity relationships of 1,3,5-alkylsubstituted cyclohexylamines binding at NMDA receptor PCP site
Wojciech Danysz
European journal of medicinal chemistry, 2000
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