Peptides derived from HIV-1 vif: a non-substrate based novel type of HIV-1 protease inhibitors 1 1 Edited by J. Karn (original) (raw)

Peptides derived from HIV-1 vif: a non-substrate based novel type of HIV-1 protease inhibitors

Chaim Gilon

Journal of Molecular Biology, 1999

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Human immunodeficiency virus type 1 Vif-derived peptides inhibit the viral protease and arrest virus production

Nissim Chen

Febs Letters, 1998

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Peptide inhibitors of HIV-1 protease and viral infection of peripheral blood lymphocytes based on HIV-1 Vif

David Volsky

Proceedings of the National Academy of Sciences, 1998

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Design, Synthesis and Screening of Novel PCU-peptide/peptoid Derived HIV Protease Inhibitors

Maya Makatini

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Abrogation of Vif function by peptide derived from the N-terminal region of the human immunodeficiency virus type 1 (HIV-1) protease

marina hutoran

Virology, 2004

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Design and synthesis of inhibitors for the HIV-1 protease

Nicholas Camp

1994

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Potency Comparison of Peptidomimetic Inhibitors against HIV-1 and HIV-2 Proteinases: Design of Equipotent Lead Compounds

Juraj Sedláček

Archives of Biochemistry and Biophysics, 1997

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An Orally Bioavailable HIV1 Protease Inhibitor Containing an Imidazole-Derived Peptide Bond Replacement: Crystallographic and Pharmacokinetic Analysis

Sherin S. Abdel-Meguid

Biochemistry, 1994

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Cyclic HIV protease inhibitors capable of displacing the active site structural water molecule

Bruce Aungst

Drug Discovery Today, 1997

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Inhibitors of HIV Protease: Unique Non‐peptide Active Site Templates

Christopher Gajda

Journal of Molecular Recognition, 1996

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Small-Molecule Inhibitors of HIV-1 Protease Dimerization Derived from Cross-Linked Interfacial Peptides

Michael Shultz

Angewandte Chemie International Edition, 2000

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Molecular Recognition of Macrocyclic Peptidomimetic Inhibitors by HIV1 Protease † , ‡

David Fairlie

Biochemistry, 1999

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Substrate-Based Cyclic Peptidomimetics of Phe-Ile-Val That Inhibit HIV-1 Protease Using a Novel Enzyme-Binding Mode

Jakob Begun

Journal of the American Chemical Society, 1996

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Future appeal of comparative studies on putative binding sites of HIV-1 virus-encoded proteolytic enzyme inhibitor of different Food and Drug Administration-approved compounds

SAMI MELEBARI

HIV & AIDS Review

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Two-step binding mechanism for HIV protease inhibitors

Thomas Spector

Biochemistry, 1992

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Pentacycloundecane derived hydroxy acid peptides: A new class of irreversible non-scissile ether bridged type isoster as potential HIV-1 wild type C-SA protease …

Yasien Sayed

Bioorganic …, 2011

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Inhibition of HIV by an anti-HIV protease synthetic peptide blocks an early step of viral replication

Jean-alain Fehrentz

Research in Virology, 1992

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Discovery and optimization of nonpeptide HIV-1 protease inhibitors

John Domagala

Bioorganic & Medicinal Chemistry, 1996

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Pentacycloundecane derived hydroxy acid peptides: A new class of irreversible non-scissile ether bridged type isoster as potential HIV-1 wild type C-SA protease inhibitors

Gert Kruger

Bioorganic Chemistry, 2012

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Development and Identification of a Novel Anti-HIV-1 Peptide Derived by Modification of the N-Terminal Domain of HIV-1 Integrase

Michele Manfra

Frontiers in Microbiology, 2016

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Structural Basis of HIV-1 and HIV-2 Protease Inhibition by a Monoclonal Antibody

J. Lescar

Structure, 2001

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Development of peptide inhibitors of HIV transmission

vivek kumar

Bioactive Materials, 2016

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Structure–activity relationship of HIV-1 protease inhibitors containing α-hydroxy-β-amino acids. Detailed study of P1 site

Shuichi Miyamoto

Bioorganic & Medicinal Chemistry, 1999

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A Novel Nonpeptide HIV-1 Protease Inhibitor: Elucidation of the Binding Mode and Its Application in the Design of Related Analogs

Donna Ferguson

Journal of Medicinal Chemistry, 1994

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Conformationally constrained HIV-1 protease inhibitors

Joseph Vacca

Bioorganic & Medicinal Chemistry Letters, 1994

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A New Generation of Peptide-based Inhibitors Targeting HIV-1 Reverse Transcriptase Conformational Flexibility

Pascal Clayette

Journal of Biological Chemistry, 2009

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Inhibition of HIV1 replication by a peptide dimerization inhibitor of HIV1 protease

Cara Brown

Antiviral Research, 2006

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Human immunodeficiency virus type 1 Vif binds the viral protease by interaction with its N-terminal region

marina hutoran

The Journal of general virology, 2002

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Antiviral agent based on the non-structural protein targeting the maturation process of HIV-1: expression and susceptibility of chimeric Vpr as a substrate for cleavage by HIV-1 protease

Irene Weber

Protein Engineering Design and Selection, 2000

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Structure of a non-peptide inhibitor complexed with HIV-1 protease. Developing a cycle of structure-based drug design

D. Decamp, Elaine Meng

The Journal of biological chemistry, 1993

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Pentacycloundecane-diol-Based HIV-1 Protease Inhibitors: Biological Screening, 2 D NMR, and Molecular Simulation Studies

Bahareh Honarparvar, Yasien Sayed

ChemMedChem, 2012

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