The synthesis, and dopamine D2 and serotonin 5-HT3 receptor affinity of 3-aza analogues (pyridyl) of 4-amino-5-chloro-2-methoxybenzamides (original) (raw)

Dopamine/Serotonin Receptor Ligands. 12 1 : SAR Studies on Hexahydro-dibenz[ d , g ]azecines Lead to 4-Chloro-7-methyl-5,6,7,8,9,14-hexahydrodibenz[ d,g ]azecin-3-ol, the First Picomolar D 5 -Selective Dopamine-Receptor Antagonist

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