original ) (raw )Dopamine/Serotonin Receptor Ligands. 10: 1 SAR Studies on Azecine-type Dopamine Receptor Ligands by Functional Screening at Human Cloned D 1 , D 2L , and D 5 Receptors with a Microplate Reader Based Calcium Assay Lead to a Novel Potent D 1 /D 5 Selective Antagonist
Sherif Rostom , Matthias Kassack , Hussein El-subbagh
Journal of Medicinal Chemistry, 2006
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Dopamine/serotonin receptor ligands. Part 17: A cross-target SAR approach: Affinities of azecine-styled ligands for 5-HT2A versus D1 and D2 receptors
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Bioorganic & Medicinal Chemistry Letters, 2008
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Dopamine/Serotonin Receptor Ligands, Part III [1]: Synthesis and Biological Activities of 7, 7′—Alkylene-bis-6, 7, 8, 9, 14, 15-hexahydro-5H-benz[d]indolo[2, 3-g]azecines — Application of the Bivalent Ligand Approach to a Novel Type of Dopamine Receptor Antagonist
Ashraf Abadi
Archiv Der Pharmazie, 2002
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Dopamine/Serotonin Receptor Ligands. Part IV [1]: Synthesis and Pharmacology of Novel 3-Benzazecines and 3-Benzazonines as Potential 5-HT2A and Dopamine Receptor Ligands
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Archiv der Pharmazie, 2002
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Synthesis and receptor affinities of some conformationally restricted analogues of the dopamine D1 selective ligand (5R)-8-chloro-2,3,4,5-tetrahydro-3-methyl-5-phenyl- 1H-3-benzazepin-7-ol
R. Chipkin , Donald Hou
Journal of medicinal chemistry, 1989
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Bioorganic & Medicinal Chemistry Letters, 2007
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Jeffrey Witkin
Journal of Medicinal Chemistry, 1995
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Val Watts
Journal of Medicinal Chemistry, 1997
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Bioorganic & Medicinal Chemistry, 2010
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Harald Hübner
Bioorganic & Medicinal Chemistry Letters, 1999
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John Neumeyer
Journal of Medicinal Chemistry, 1991
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Jeffrey Witkin
Journal of Medicinal Chemistry, 1996
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Structure−Activity Relationships for a Novel Series of Dopamine D2-like Receptor Ligands Based on N-Substituted 3-Aryl-8-azabicyclo[3.2.1]octan-3-ol
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Journal of Medicinal Chemistry, 2008
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Archiv Der Pharmazie, 2021
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Frank King
Bioorganic & Medicinal Chemistry Letters, 1995
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Richard Mailman
European Journal of Pharmacology, 1993
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Ferran Sanz
Bioorganic & Medicinal Chemistry Letters, 2009
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martyn wood
Bioorganic & Medicinal Chemistry Letters, 2000
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Ross Baldessarini
Drug Discovery Today, 1997
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Vicki COFFIN
Bioorganic & Medicinal Chemistry Letters, 1992
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Michael Wiese
BMC pharmacology, 2006
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Charles Ashby
Journal of Medicinal Chemistry, 2010
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trans-2,6-, 3,6- and 4,6-Diaza-5,6,6a,7,8,12b-hexahydrobenzo[C]phenanthrene-10,11-diols as dopamine agonists
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Bioorganic & Medicinal Chemistry Letters, 1999
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Bioorganic & Medicinal Chemistry, 2013
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Anna C Cunha
Bioorganic & Medicinal Chemistry, 2003
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Bioorganic & Medicinal Chemistry Letters, 2006
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Bioorganic & Medicinal Chemistry Letters, 2010
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Bioorganic & Medicinal Chemistry Letters, 1998
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Dopamine receptor agonists: 3-allyl-6-chloro-2,3,4,5-tetrahydro-1-(4-hydroxyphenyl)-1H-3-benzazepine-7,8-diol and a series of related 3-benzazepines
Robert Demarinis
Journal of Medicinal Chemistry, 1986
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