Stimulation of bone formation and prevention of bone loss by prostaglandin E EP4 receptor activation (original) (raw)

The Role of Prostaglandin E Receptor Subtypes (EP1, EP2, EP3, and EP4) in Bone Resorption: An Analysis Using Specific Agonists for the Respective EPs

Yukihiko Sugimoto

Endocrinology, 2000

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Impaired Bone Resorption to Prostaglandin E2 in Prostaglandin E Receptor EP4-knockout Mice

Yukihiko Sugimoto

Journal of Biological Chemistry, 2000

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Prostaglandin Receptor EP4Mediates the Bone Anabolic Effects of PGE2

Michel Gallant

Molecular Pharmacology, 2001

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Prostaglandin E2 Directly Inhibits Bone-Resorbing Activity of Isolated Mature Osteoclasts Mainly Through the EP4 Receptor

M MANO

Calcified Tissue International, 2000

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A Nonprostanoid EP4 Receptor Selective Prostaglandin E2 Agonist Restores Bone Mass and Strength in Aged, Ovariectomized Rats

Kimberly Cameron

Journal of Bone and Mineral Research, 2005

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Systemic prostaglandin E2 increases cancellous bone formation and mass in aging rats and stimulates their bone marrow osteogenic capacity in vivo and in vitro

S. Keila

Journal of Endocrinology, 2001

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Impaired Bone Resorption by Lipopolysaccharide In Vivo in Mice Deficient in the Prostaglandin E Receptor EP4 Subtype

Yukihiko Sugimoto

Infection and Immunity, 2000

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Prostaglandin E2 (PGE2) increases the number of rat bone marrow osteogenic stromal cells (BMSC) via binding the EP4 receptor, activating sphingosine kinase and inhibiting caspase activity

S. Keila

Prostaglandins, Leukotrienes and Essential Fatty Acids, 2006

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Discovery of CP533536: An EP 2 receptor selective prostaglandin E 2 (PGE 2) agonist that induces local bone formation

christina wright

Bioorganic & Medicinal Chemistry Letters, 2009

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Augmentation of bone morphogenetic protein-induced bone mass by local delivery of a prostaglandin E EP4 receptor agonist

Hidetomi Terai

Bone, 2005

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A prostanoid receptor EP4 agonist enhances ectopic bone formation induced by recombinant human bone morphogenetic protein-2

Hidetomi Terai

Biochemical and Biophysical Research Communications, 2004

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An EP2 receptor-selective prostaglandin E2 agonist induces bone healing

Bruce Lefker

Proceedings of the National Academy of Sciences, 2003

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Immunolocalization of the prostaglandin E2 receptor subtypes in human bone tissue: differences in foetal, adult normal, osteoporotic and pagetic bone

A. Brum-fernandes

Prostaglandins, Leukotrienes and Essential Fatty Acids, 2004

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Prostaglandin E 2 Strongly Inhibits Human Osteoclast Formation

Nobuyuki Udagawa

Endocrinology, 2005

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A Novel, Non-Prostanoid EP2 Receptor-Selective Prostaglandin E2 Agonist Stimulates Local Bone Formation and Enhances Fracture Healing

Bruce Lefker

Journal of Bone and Mineral Research, 2003

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Inhibitory and stimulatory effects of prostaglandins on osteoclast differentiation

Afsie Sabokbar

Calcified Tissue International, 1997

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Prostaglandin E2 receptor (EP4) selective agonist (ONO-4819.CD) accelerates bone repair of femoral cortex after drill-hole injury associated with local upregulation of bone turnover in mature rats

Toshitaka Nakamura

Bone, 2004

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Effects of Basic Fibroblast Growth Factor and a Prostaglandin E2 Receptor Subtype 4 Agonist on Osteoblastogenesis and Adipogenesis in Aged Ovariectomized Rats

Marda Jorgensen

Journal of Bone and Mineral Research, 2007

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Systemic administration of an anabolic dose of PGE2 in young rats increases the osteogenic capacity of bone marrow

S. Keila

Bone, 1997

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Prostaglandin EP4 Selective Agonist AKDS001 Enhances New Bone Formation by Minimodeling in a Rat Heterotopic Xenograft Model of Human Bone

Zeynep Bal

Frontiers in Bioengineering and Biotechnology, 2022

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Effects of prostaglandins on rat calvarial bone-cell calcium

Rosemary Dziak

Archives of Oral Biology, 1984

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Discovery of highly selective EP4 receptor agonists that stimulate new bone formation and restore bone mass in ovariectomized rats

Margaret Chu-Moyer, Michael Zawistoski, Bruce Lefker, Kimberly Cameron

Bioorganic & Medicinal Chemistry Letters, 2006

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Prostaglandin E2 Stimulates Fibronectin Expression through EP1 Receptor, Phospholipase C, Protein Kinase Cα, and c-Src Pathway in Primary Cultured Rat Osteoblasts

Rong-sen Yang

Journal of Biological Chemistry, 2005

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Osteoblasts Are a New Target for Prolactin: Analysis of Bone Formation in Prolactin Receptor Knockout Mice 1

Brigitte Bouchard, Philippe Clément-lacroix

Endocrinology, 1999

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Osteoblasts are a new target for prolactin: Analysis of bone formation in prolactin receptor knockout mice

Vincent Goffin

Endocrinology

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Novel EP4 receptor agonist-bisphosphonate conjugate drug (C1) promotes bone formation and improves vertebral mechanical properties in the ovariectomized rat model of postmenopausal bone loss

JOHN GEORGIOU

Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2014

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Lights and shadows of NSAIDs in bone healing: the role of prostaglandins in bone metabolism

Karolina Domaracka

Drug Design Development and Therapy, 2018

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Systemic effects of prostaglandin E2 on vertebral trabecular remodeling in beagles used in a healing study

Mei-Shu Shih

Calcified Tissue International, 1988

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Characterization of the prostaglandin receptors in human osteoblasts in culture

Ghassan Bkaily

Prostaglandins, Leukotrienes and Essential Fatty Acids, 2001

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Regulation of bone biology by prostaglandin endoperoxide H synthases (PGHS): A rose by any other name…

Allison Pettit

Cytokine & Growth Factor Reviews, 2006

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Prostaglandin G/H synthase-2 is required for maximal formation of osteoclast-like cells in culture

Scott Morham

Journal of Clinical Investigation, 2000

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Prostaglandin E2 enhances alveolar bone formation in the rat mandible

Laurence Walsh

Bone, 2004

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Inactivation of estrogen receptor in bone-forming cells induces bone loss in female mice

kalman buki

The FASEB Journal, 2013

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Osteopontin deficiency enhances anabolic action of EP4 agonist at a sub-optimal dose in bone

Jono Yang

Journal of Endocrinology, 2007

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