Matrix metalloproteinase–activated doxorubicin prodrugs inhibit HT1080 xenograft growth better than doxorubicin with less toxicity (original) (raw)

Matrix metalloproteinase-activated doxorubicin prodrugs inhibit HT1080 xenograft growth better than …

Daniel Hu

Molecular cancer therapeutics

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Discovery of matrix metalloproteases selective and activated peptide–doxorubicin prodrugs as anti-tumor agents

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A New Approach for the Treatment of Malignant Melanoma: Enhanced Antitumor Efficacy of an Albumin-binding Doxorubicin Prodrug That Is Cleaved by Matrix Metalloproteinase 21

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2000

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A new approach for the treatment of malignant melanoma: enhanced antitumor efficacy of an albumin-binding doxorubicin prodrug that is cleaved by matrix metalloproteinase 2

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Paradoxical Stimulation of Matrix Metalloproteinase-9 Expression in HT1080 Cells by a Broad-Spectrum Hydroxamate-Based Matrix Metalloproteinase Inhibitor

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Development of matrix metalloproteinase inhibitors in cancer therapy

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New approaches to selectively target cancer-associated matrix metalloproteinase activity

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Critical appraisal of the use of matrix metalloproteinase inhibitors in cancer treatment

Wen-Tien Chen

Oncogene, 2000

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Inhibition of metalloproteinases derived from tumours: New insights in the treatment of human glioblastoma

Elisa Nuti, Elisabetta Orlandini, Armando Rossello

2010

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Matrix-metalloproteinases as targets for controlled delivery in cancer: An analysis of upregulation and expression

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A matrix metalloproteinase 2 cleavable melittin/avidin conjugate specifically targets tumor cells in vitro and in vivo

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International Journal of Oncology, 2003

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Tumour microenvironment — Opinion: Validating matrix metalloproteinases as drug targets and anti-targets for cancer therapy

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Nature Reviews Cancer, 2006

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Matrix metalloproteinase and its drug targets therapy in solid and hematological malignancies: An overview

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Mutation Research/Reviews in Mutation Research, 2013

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Anticancer activity of PEGylated matrix metalloproteinase cleavable peptide-conjugated adriamycin against malignant glioma cells

Young-Il Jeong

International journal of pharmaceutics, 2010

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Matrix Metalloproteinase Inhibitors as Anticancer Therapeutics

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Current Cancer Drug Targets, 2005

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Stimulation of Matrix Metalloproteinase-9 Expression in Human Fibrosarcoma Cells by Synthetic Matrix Metalloproteinase Inhibitors

Charles Lambert, Carine Munaut

Experimental Cell Research, 2002

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A phase I dose escalation study of the matrix metalloproteinase inhibitor BAY 12-9566 administered orally in patients with advanced solid tumours

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Annals of oncology : official journal of the European Society for Medical Oncology / ESMO, 2000

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Small-molecule anticancer compounds selectively target the hemopexin domain of matrix metalloproteinase-9

CEM KUSCU

Cancer research, 2011

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Anti-Invasive, Antitumoral, and Antiangiogenic Efficacy of a Pyrimidine-2,4,6-trione Derivative, an Orally Active and Selective Matrix Metalloproteinases Inhibitor

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Clinical Cancer Research, 2004

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Inhibition of Angiogenesis and Metastasis In Two Murine Models by the Matrix Metalloproteinase Inhibitor, BMS-275291

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Ensnaring membrane type 1-matrix metalloproteinase (MT1-MMP) with tissue inhibitor of metalloproteinase (TIMP)-2 using the haemopexin domain of the protease as a carrier: a targeted approach in cancer inhibition

Huee Lee

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In Vitro Efficacy of a Sterically Stabilized Immunoliposomes Targeted to Membrane Type 1 Matrix Metalloproteinase (MT1-MMP)

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Biological & Pharmaceutical Bulletin, 2007

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Matrix metalloproteinase inhibitors: Applications in oncology

D. Yip

Investigational New Drugs, 1999

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A novel and selective membrane type-1 matrix metalloproteinase (MT1-MMP) inhibitor reduces cancer cell motility and tumor growth

Tuula Salo

Cancer Biology & Therapy, 2009

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Data from Selective Inhibition of Matrix Metalloproteinase-14 Blocks Tumor Growth, Invasion, and Angiogenesis

nicolas frans

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Selective Inhibition of Matrix Metalloproteinase-14 Blocks Tumor Growth, Invasion, and Angiogenesis

nicolas frans

Cancer Research, 2009

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Modulation of Tumor Cell Growth In Vivo by Extracellular Matrix Metalloprotease Inducer

William Grizzle

Archives of Otolaryngology–Head & Neck Surgery, 2008

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CD10 is a key enzyme involved in the activation of tumor-activated peptide prodrug CPI-0004Na and novel analogues: implications for the design of novel peptide prodrugs for the therapy of CD10+ tumors

Dana Buckman

Cancer research, 2003

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Matrix metalloprotease selective peptide substrates cleavage within hydrogel matrices for cancer chemotherapy activation

Syed Salman Lateef

Peptides, 2008

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Matrix metalloproteinases in cancer: from new functions to improved inhibition strategies

luis sanchez

International Journal of Developmental Biology, 2004

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Functional Analysis of Matrix Metalloproteinases and Tissue Inhibitors of Metalloproteinases Differentially Expressed by Variants of Human HT-1080 Fibrosarcoma Exhibiting High and Low Levels of Intravasation and Metastasis

Elena Deryugina

Journal of Biological Chemistry, 2007

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