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Journal of Medicinal Chemistry, 1997
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Pure and Applied Chemistry, 2000
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New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
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Bioorganic & Medicinal Chemistry Letters, 2006
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Synthesis of 7,8-(Methylenedioxy)-1-phenyl-3,5-dihydro-4 H -2,3-benzodiazepin- 4-ones as Novel and Potent Noncompetitive AMPA Receptor Antagonists
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Journal of Medicinal Chemistry, 1998
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New Insight into the Central Benzodiazepine Receptor–Ligand Interactions: Design, Synthesis, Biological Evaluation, and Molecular Modeling of 3-Substituted 6-Phenyl-4 H -imidazo[1,5- a ][1,4]benzodiazepines and Related Compounds
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Journal of Medicinal Chemistry, 2011
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Activity of 2,3-benzodiazepines at Native Rat and Recombinant Human Glutamate Receptors In Vitro: Stereospecificity and Selectivity Profiles
István Tarnawa
Neuropharmacology, 1996
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Specific inhibition of benzodiazepine receptor binding by some N-(indol-3-ylglyoxylyl)amino acid derivatives
G. Biagi
Journal of Medicinal Chemistry, 1985
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6-(4-Pyridinyl)-1H-1,2,3-triazolo[4,5-d]-pyrimidin-4(5H)-one: A Structurally Novel Competitive AMPA Receptor Antagonist
balbir B singh, Adi Treasurywala
Journal of Medicinal Chemistry, 1995
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Recent Structure Activity Relationship Studies of 1,4-Benzodiazepines
Peertechz Journals
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New non competitive AMPA antagonists
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Bioorganic & Medicinal Chemistry, 2000
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Computer-aided investigation of the structure–activity relationships of benzodiazepine derivatives at diazepam-sensitive receptors
Anatoli Dimoglo
Journal of Molecular Structure-theochem, 1999
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Synthesis, Chiral Resolution, and Enantiopharmacology of a Potent 2,3Benzodiazepine Derivative as Noncompetitive AMPA Receptor Antagonist
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Journal of Medicinal Chemistry, 2006
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Synthesis and characterization of 8-ethynyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one derivatives: Part 2. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists
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Bioorganic & Medicinal Chemistry Letters, 2008
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Synthesis and Evaluation of Pharmacological Properties of Novel Annelated 2,3-Benzodiazepine Derivatives
Giovambattista Sarro
Journal of Medicinal Chemistry, 2003
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An Updated Unified Pharmacophore Model of the Benzodiazepine Binding Site on γ-Aminobutyric Acida Receptors: Correlation with Comparative Models
Craig Morton
Current Medicinal Chemistry, 2007
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Search for Structural Requirements of 2–Phenylimidazo [1, 2–α] pyridineacetamide Analogs to Improve Affinity and Selectivity towards Central and/or Peripheral Benzodiazepine Receptors
Tarun Jha
2007
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Phthalazine-1,4-dione derivatives as non-competitive AMPA receptor antagonists: design, synthesis, anticonvulsant evaluation, ADMET profile and molecular docking
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Molecular Diversity, 2018
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Molecular modeling studies, synthesis, configurational stability and biological activity of 8-chloro-2,3,5,6-tetrahydro-3,6-dimethyl-pyrrolo[1,2,3-de]-1,2,4-benzothiadiazine 1,1-dioxide
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Bioorganic & Medicinal Chemistry, 2011
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Search for Structural Requirements of 2–Phenylimidazo[1,2–] pyridineacetamide Analogs to Improve Affinity and Selectivity towards Central and/or Peripheral Benzodiazepine Receptors
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Internet Electronic Journal of Molecular Design, 2007
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Functional characterization of CP-465,022, a selective, noncompetitive AMPA receptor antagonist
Fiona Ewing
Neuropharmacology, 2002
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Studies on specific inhibition of benzodiazepine receptor binding by some C-benzoyl-1,2,3-triazole derivatives
G. Biagi
Journal of Pharmaceutical Sciences, 1993
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Synthesis and anticonvulsant activity of N-3 substituted 2,3-benzodiazepines
Giovambattista Sarro
Il Farmaco, 2004
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Mapping the Peripheral Benzodiazepine Receptor Binding Site by Conformationally Restrained Derivatives of 1-(2-Chlorophenyl)- N -methyl- N -(1-methylpropyl)-3-isoquinolinecarboxamide (PK11195)
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Journal of Medicinal Chemistry, 1997
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Analogs of 3-Hydroxy-1 H- 1-benzazepine-2,5-dione: Structure−Activity Relationship at N -Methyl- d -aspartate Receptor Glycine Sites
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J Med Chem, 1996
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7-Chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine S,S-dioxide: A partial modulator of AMPA receptor desensitization devoid of neurotoxicity
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Proceedings of the National Academy of Sciences, 1997
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New 3-, 8-disubstituted pyrazolo[5,1-c][1,2,4]benzotriazines useful for studying the interaction with the HBp-3 area (hydrogen bond point area) in the benzodiazepine site on the γ-aminobutyric acid type A (GABAA) receptor
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Bioorganic & Medicinal Chemistry, 2011
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Characterization of the 1H-Cyclopentapyrimidine-2,4(1H,3H)-dione Derivative (S)-CPW399 as a Novel, Potent, and Subtype-Selective AMPA Receptor Full Agonist with Partial Desensitization Properties
anna ramunno
Journal of Medicinal Chemistry, 2001
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